Publications

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Publications

2024
Asymmetric, Remote C(sp(3) )-H Arylation via Sulfinyl-Smiles Rearrangement.
Angew Chem Int Ed Engl. 2024, e202319158
Visible Light-Mediated Heterodifunctionalization of Alkynylazobenzenes for 2H-Indazole Synthesis.
Org Lett. 2024, 26, 1868
Plaza 3055
Advanced Synthesis & Catalysis. 2024; 366(2):232 -240.
Chiral arylsulfinylamides as reagents for visible light-mediated asymmetric alkene aminoarylations.
Nat Chem. 2024, s41557-023-01414-8.

2023
1,2,3-Benzotriazine Synthesis by Heterocyclization of p-Tosylmethyl Isocyanide Derivatives.
The Journal of Organic Chemistry. 2023; 88(19):14131 -14139.
Visible-light mediated synthesis of bicalutamide by regioselective hydroxysulfonylation of acrylamides.
European Journal of Organic Chemistry. 2023; n/a(n/a):e202300535.
One-Pot (3 + 2) Cycloaddition-Isomerization-Oxidation of 2,2,2-Trifluorodiazoethane and Styryl Derivatives.
J Org Chem. 2023, doi: 10.1021/acs.joc.3c00396.
Hyper-Cross-Linked Porous Polymer Featuring B-N Covalent Bonds (HCP-BNs): A Stable and Efficient Metal-Free Heterogeneous Photocatalyst.
ACS Macro Lett. 2023, 12(7):949-954. doi: 10.1021/acsmacrolett.3c00217. Epub 2023 Jun 29.
β-Functionalization of 4 a-aza-8 a-boranaphthalene via Iridium-catalyzed C−H Borylation.
Advanced Synthesis & Catalysis. 2023; n/a(n/a).
Mizoroki-Heck Macrocyclization Reactions at 1 M Concentration Catalyzed by Sub-nanometric Palladium Clusters.
ChemSusChem. 2023; n/a(n/a):e202300200.
Visible-Light-Mediated Regioselective Chlorosulfonylation of Acrylamides.
2023; (EFirst).
Gold-catalyzed endo-selective cyclization of alkynylcyclobutanecarboxamides: synthesis of cyclobutane-fused dihydropyridones.
Org Biomol Chem. 2023,21,2705-2708. doi: 10.1039/d3ob00051f.
Synthesis of Five-Membered Organoborate Heterocycles via a Metal-Free Carboboration and Their Use in Cross-Coupling Reactions.
2023; (EFirst).

2022
Synthesis of Phenanthrene-Based Polycycles by Gold(I)-Catalyzed Cyclization of Biphenyl-Embedded Trienynes.
Advanced Synthesis & Catalysis. 2022; n/a(n/a).
Gold(I) Catalysis Applied to the Stereoselective Synthesis of Indeno%2,1-b%thiochromene Derivatives and Seleno Analogues.
Organic Letters. 2022;.
Highly efficient unbridged D-A+(D) chromophores based on the quinolizinium cation for nonlinear optical (NLO) applications.
2022; 205:110323.
Synthesis of BN-Polyarenes by a Mild Borylative Cyclization Cascade.
Org Lett. 2022;24(31):5860-5865. doi: 10.1021/acs.orglett.2c02477.
Steviol glycosides as an alternative osmotic agent for peritoneal dialysis fluid.
Front Pharmacol. 2022 Aug 16;13:868374. doi: 10.3389/fphar.2022.868374. eCollection 2022.
Synthesis of Tri- and Tetrasubstituted Alkenyl Boronates from Alkynes.
European Journal of Organic Chemistry. 2022; 2022(30):e202200521.
Insight into the mechanism of molecular recognition between human Integrin-Linked Kinase and Cpd22 and its implication at atomic level.
J Comput Aided Mol Des. 2022 Aug;36(8):575-589. doi: 10.1007/s10822-022-00466-1.
Metal-Free Temperature-Controlled Regiodivergent Borylative Cyclizations of Enynes: BCl(3) -Promoted Skeletal Rearrangement.
Angew Chem Int Ed Engl. 2022 May 5:e202205651. doi: 10.1002/anie.202205651.
Electrochemically driven one-pot oxidative conversion of arylhydrazines into aromatic iodides.
2022; 10(3):107486.
RICORS2040: the need for collaborative research in chronic kidney disease.
Clin Kidney J. 2021 Sep 23;15(3):372-387. doi: 10.1093/ckj/sfab170. eCollection 2022 Mar.
CKD: The burden of disease invisible to research funders.
Nefrologia. 2022, 42, 65
Pyridazino-pyrrolo-quinoxalinium salts as highly potent and selective leishmanicidal agents targeting trypanothione reductase.
Eur J Med Chem. 2022, 227, 113915

2021
1,10a-Dihydro-1-aza-10a-boraphenanthrene and 6a,7-Dihydro-7-aza-6a-boratetraphene: Two New Fluorescent BN-PAHs.
J. Org. Chem. 2021, 86, 23, 16259
Two-photon activated precision molecular photosensitizer targeting mitochondria.
Commun Chem 2021, 4, 142
A Computer-Driven Scaffold-Hopping Approach Generating New PTP1B Inhibitors from the Pyrrolo%1,2-a%quinoxaline Core.
ChemMedChem. 2021, 16, 2895
Chemical recovery of waste electrical and electronic equipment by microwave-assisted pyrolysis: A review.
J Anal Appl Pyrolysis 2021, 159, 105323
Enantioselective Copper-Catalyzed Synthesis of Trifluoromethyl-Cyclopropylboronates.
Org Lett. 2021, 23, 6174
Pyrrolo%1,2-a%quinoxal-5-inium salts and 4,5-dihydropyrrolo%1,2-a%quinoxalines: Synthesis, activity and computational docking for protein tyrosine phosphatase 1B.
Bioorg Med Chem. 2021, 44, 116295
Tripeptides as Integrin-Linked Kinase Modulating Agents Based on a Protein-Protein Interaction with α-Parvin.
ACS Med Chem Lett. 2021, 12, 1656
Recent developments in the chemistry of BN-aromatic hydrocarbons.
Adv. Heterocycl. Chem. 2021, 197
A new family of fluorescent pyridazinobenzimidazolium cations with DNA binding properties.
Dyes Pigm. 2021, 192, 109443
Asymmetric, visible light-mediated radical sulfinyl-Smiles rearrangement to access all-carbon quaternary stereocentres.
Nat Chem. 2021, 13, 327

2020
Selective Synthesis of Phenanthrenes and Dihydrophenanthrenes via Gold-Catalyzed Cycloisomerization of Biphenyl Embedded Trienynes.
Org Lett. 2020, 22, 8464
Gold-Catalyzed Synthetic Strategies towards Four-Carbon Ring Systems.
Catalysts 2020, 22, 1178
Pyrrolo%@5B1,2-a%@5Dquinoxalines: Insulin Mimetics that Exhibit Potent and Selective Inhibition against Protein Tyrosine Phosphatase 1B.
ChemMedChem 2020, 15, 1788
The pHLIP system as a vehicle for microRNAs in the kidney.
Nefrologia. 2020, 40, 491
Practical Solvent-Free Microwave-Assisted Hydroboration of Alkynes.
Eur. J. Org. Chem. 2020, 3024
Expanding the BN-embedded PAH family: 4a-aza-12a-borachrysene.
Chem Commun 2020, 56, 3669
Synthesis and Photophysical Behavior of a Highly Fluorescent Family of Unsymmetrical Organoboron Complexes Containing 5-(Pyridin-2-ylmethylene)imidazolidine-2,4-dione Moieties.
J Org Chem. 2020, 85, 441

2019
A New Member of the BN-Phenanthrene Family: Understanding the Role of the B-N Bond Position.
J Org Chem. 2019, 84, 7113
Remarkable effect of alkynyl substituents on the fluorescence properties of a BN-phenanthrene.
Beilstein J. Org. Chem. 2019, 15, 1257
NIK as a Druggable Mediator of Tissue Injury.
Trends Mol Med. 2019, 25, 341
Synthesis, Functionalization, and Optical Properties of 1,2-Dihydro-1-aza-2-boraphenanthrene and Several Highly Fluorescent Derivatives.
Org Lett. 2019, 21, 2550
Regiodivergent Electrophilic Cyclizations of Alkynylcyclobutanes for the Synthesis of Cyclobutane-Fused O-Heterocycles.
J. Org. Chem. 2019, 84, 9, 5712
MAP3K kinases and kidney injury.
Nefrologia 2019, 39, 568

2018
Discovery of potent calpain inhibitors based on the azolo-imidazolidenone.
Eur J Med Chem. 2018, 157, 946
C-H Functionalization of BN-Aromatics Promoted by Addition of Organolithium Compounds to the Boron Atom.
Org Lett. 2018, 20, 4902
gamma-Carboline Synthesis by Heterocyclization of TosMIC Derivatives.
J Org Chem. 2018, 83, 6623
A Tricin Derivative from Deschampsia antarctica Desv. Inhibits Colorectal Carcinoma Growth and Liver Metastasis through the Induction of a Specific Immune Response.
Mol Cancer Ther. 2018 May;17(5):966-976. doi: 10.1158/1535-7163.MCT-17-0193. Epub 2018 Feb 26.
Dibenzopyridoimidazocinnolinium cations: a new family of light-up fluorescent DNA probes.
Org. Chem. Front. 2018, 5, 1916
Synthesis of functionalized helical BN-benzo%c%phenanthrenes.
Chem Commun 2018, 54, 2467

2017
Azonia aromatic heterocycles as a new acceptor unit in D-π-A%@2B vs D-A%@2B nonlinear optical chromophores.
Dyes Pigm. 2017, 144, 17
Microwave-assisted pyrolysis of Mediterranean forest biomass waste: Bioproduct characterization.
J Anal Appl Pyrolysis 2017, 127, 278
Synthesis, Optical Properties, and Regioselective Functionalization of 4a-Aza-10a-boraphenanthrene.
Org Lett. 2017, 19, 3458
Imidazopyridinium cations: A new family of azonia aromatic heterocycles with applications as DNA intercalators.
Dyes Pigm. 2017, 138, 135
Quinolizinium as a new fluorescent lysosomotropic probe.
Biorg. Med. Chem. Lett. 2017, 27, 203
Halogen-containing thiazole orange analogues - new fluorogenic DNA stains.
Beilstein J. Org. Chem. 2017, 13, 2902

2016
Recent Advances in the Synthesis of Azonia Aromatic Heterocycles.
J Org Chem. 2016, 81, 10126
Synthesis of 1-Substituted Isoquinolines by Heterocyclization of TosMIC Derivatives: Total Synthesis of Cassiarin A.
Org Lett. 2016, 18, 3378

2015
Highly Fluorescent Green Fluorescent Protein Chromophore Analogues Made by Decorating the Imidazolone Ring.
Chem. Eur. J. 2015, 21, 18758
Assembly of New Merocyanine Chromophores with a 1,8-Naphthalimide Core by a New Method for the Synthesis of the Methine Function.
Aust. J. Chem. 2015, 68, 1399
Nonlinear Emission of Quinolizinium Based Dyes With Application in Fluorescence Lifetime Imaging.
J. Phys. Chem. A 2015, 119, 11, 2351
Azonia Aromatic Cations by Ring-Closing Metathesis: Synthesis ofAzaquinolizinium Cations.
Eur J Org Chem. 2015, 6, 4214
Synthesis and biological evaluation of pyridazino%@5B1′,6′:1,2%@5Dpyrido%@5B3,4-b%@5Dindolinium and pyridazino%@5B1,6-a%@5Dbenzimidazolium salts as anti-inflammatory agents.
Eur. J. Med. Chem. 2015, 93, 83
Isoquinoline synthesis by heterocyclization of tosylmethyl isocyanide derivatives: total synthesis of mansouramycin B.
Org Lett. 2015, 17, 78
Targeting DNA with small molecules: a comparative study of a library of azonia aromatic chromophores.
Org Biomol Chem. 2015, 13, 527

2014
Efficient synthesis of an indoloquinolizinium alkaloid selective DNA-binder by ring-closing metathesis.
Org Lett. 2014, 16, 3464
Microwave-assisted synthesis of potent PDE7 inhibitors containing a thienopyrimidin-4-amine scaffold.
Org Biomol Chem. 2014, 12, 4233
Cucurbit%n%urils as a potential fine-tuned instrument for modifying photophysical properties of D–π–A+–π–D “push–pull” chromophores.
Dyes Pigm. 2014, 103, 106
Novel charged NLO chromophores based on quinolizinium acceptor units.
Dyes Pigm. 2014, 101, 116

2013
Remote aryl cyanation via isocyanide-cyanide rearrangement on tosylmethyl isocyanide derivatives.
Org Lett. 2013, 15, 3388
Synthesis of charged bis-heteroaryl donor-acceptor (D-A+) NLO-phores coupling (π-deficient-π-excessive) heteroaromatic rings.
Org. Biomol. Chem. 2013, 11, 7145
Fluorescent Dyes for Bio-Applications in the Patent Literature / Fluorescent Dyes for Bio-Applications in the Patent Literature
Current Materials Science. 2013; 6(2):81 -119. doi: 10.2174/1874464811306020001
Synthesis and evaluation of quinazoline derivatives as phosphodiesterase 7 inhibitors.
Bioorg. Med. Chem. 2013, 21, 2370

2012
A cascade reaction of azolopyrimidines. Synthesis of unusual indole and azaindole derivatives.
Chem. Commun. 2012, 48, 9171
Donor-(π-bridge)-azinium as D-π-A + one-dimensional and D-π-A +-π-D multidimensional V-shaped chromophores.
Org. Biomol. Chem. 2012, 10, 1659
Superior Neuroprotective Efficacy of LAU-0901, a Novel Platelet-Activating Factor Antagonist, in Experimental Stroke.
Translational Stroke Research 2012, 3, 154
Synthesis of 9,9′-%1,2-Ethanediylbis(oxymethylene)%bis-2-amino-1,9-dihydro-6H-purin-6-one, an Impurity of Acyclovir.
Molecules 2012, 17, 8735
New losartan-hydrocaffeic acid hybrids as antihypertensive-antioxidant dual drugs: Ester, amide and amine linkers
Eur. J. Med. Chem 2012, 50, 90

2011
A V-shaped cationic dye for nonlinear optical bioimaging.
Chem. Commun. 2011, 47, 7374
Radical Intramolecular Arylation of Pyridinium Salts: A Straightforward Entry to 7-Hydroxypyrido%2,1‐a%isoquinolinylium Salts /
Eur. J. Org. Chem. 2011, 619
Ethyl 4,4-dimethyl pyroglutamate (DMPG): A chiral auxiliary in cyclopropanation and carbonyl group activator.
Arkivoc 2011, 3, 42
Novel linear and V-shaped D-π-A+-π-D chromophores by Sonogashira reaction.
Arkivoc 2011, 3, 140
An environmentally benign procedure for the synthesis of substituted 2-thiobenzothiazoles, 2-thiobenzoxazoles, 2-thiobenzimidazoles, and 1,3-oxazolopyridine-2-thiols.
Monatsh. Chem. 2011, 142, 895
Synthesis of novel tetracationic asymmetric monomeric monomethine cyanine dyes – highly fluorescent dsDNA probes /
Coloration Technology. 2011, 127, 69
Environmental Risk Assessment of Emerging Pollutants in Water: Approaches Under Horizontal and Vertical EU Legislation /
Critical Reviews in Environmental Science and Technology 2011, 41, 699
Ring-Closing Metathesis Approach to Heteroaromatic Cations: Synthesis of Benzo%a%Dquinolizinium Salts /
Eur. J. Org. Chem. 2011, 1280

2010
Heteroaromatic Cation-Based Chromophores: Synthesis and Nonlinear Optical Properties of Alkynylazinium Salts /
Eur. J. Org. Chem. 2010, 6323
Application of Selective Palladium-Mediated Functionalization of the Pyrido%@5B3′,2′:4,5%@5Dpyrrolo%@5B1,2-c%@5Dpyrimidine Heterocyclic System for the Total Synthesis of Variolin B and Deoxyvariolin B /
Eur. J. Org. Chem. 2010, 5607
Novel Green Procedure for the Synthesis of 2-Arylbenzothiazoles Under Microwave Irradiation in Peg 200 Or Peg 400 /
Phosphorus, Sulfur, and Silicon and the Related Elements 2010, 185, 2292
Styryl dyes – synthesis and applications during the last 15 years /
Coloration Technology. 2010, 126, 55
Green chemistry in organic synthesis.
Mini-Reviews in Organic Chemistry. 2010, 7, 44
Novel environmentally benign procedure for the synthesis of 2-aryl- and 2-hetaryl-4(3H)-quinazolinones /
Coloration Technology 2010, 126, 24
An easy and fast ultrasonic selective S-alkylation of hetaryl thiols at room temperature /
Ultrasonics Sonochemistry 2010, 17, 783

Topics ...
Publications